Profile: MedKoo Biosciences is a provider of drug molecules and drug agents. We offer many active pharmaceutical ingredients and drug intermediates. Our API drugs include adapalene, adefovir dipivoxil, bicalutamide, dimecrotic acid, eperisone hydrochloride, lafutidine, levetiracetam, olmesartan, lomefloxacin monohydrochloride, pidotimod, risperidone, roxatidine acetate and rizatriptan benzoate. Our drug intermediates include adapalene, bicalutamide, escitalopram, olmesartan, pioglitazone, sumatriptan, temozolomide, pazufloxacin, liranaftate and zolmitriptan. We provide services such as collaboration research and contract organic synthesis, which include early stage discovery needs, medicinal & process chemistry. We offer products and service from discovery and early medicinal chemistry to multiple kilogram scale synthesis. Our research services include medicinal chemistry research, custom organic synthesis, synthetic route optimization, synthetic process development, formulation development and bioanalytical services. Our molecular building blocks are used for chemical modification of a lead molecule so as to enhance the potency, to reduce the side-effects, to improve oral bioavailability, and to increase aqueous solubility.
• Nolatrexed
IUPAC Name: 2-amino-6-methyl-5-pyridin-4-ylsulfanyl-1H-quinazolin-4-one | CAS Registry Number: 147149-76-6 Synonyms: Nolatrexed [INN], AIDS157719, AIDS-157719, CID108189, NCGC00181023-01, NCI60_016753, NSC648316 (HYDROCHLORIDE SALT), LS-187627, 2-Amino-6-methyl-5-(4-pyridylthio)-4(3H)-quinazolinone., 2-Amino-6-methyl-5-(4-pyridinylthio)-4-quinazolinol hydrochloride
InChIKey: XHWRWCSCBDLOLM-UHFFFAOYSA-N | ||||||||
• Noscapine Base
IUPAC Name: (3S)-6,7-dimethoxy-3-[(5R)-4-methoxy-6-methyl-7,8-dihydro-5H-[1,3]dioxolo[4,5-g]isoquinolin-5-yl]-3H-2-benzofuran-1-one | CAS Registry Number: 128-62-1 Synonyms: noscapine, alpha-Narcotine, Narcompren, Tusscapine, Narcosine, Noscopine, Terbenol, Opianin, Capval, .beta.-Narcotine, Noscapine (TN), (S,R)-Noscapine, Prestwick_959, NARCOTINE, Noscapine hydrchloride, Tocris-1697, Coscopin;Methoxyhydrastine, Prestwick0_000563, Prestwick1_000563, Prestwick2_000563
InChIKey: AKNNEGZIBPJZJG-MSOLQXFVSA-N | ||||||||
• Oxiracetam
IUPAC Name: 2-(4-hydroxy-2-oxopyrrolidin-1-yl)acetamide | CAS Registry Number: 62613-82-5 Synonyms: oxiracetam, Hydroxypiracetam, Neuractiv, Neuromet, Oriest, 4-Hydroxypiracetam, (+-)-Oxiracetam, Oxiracetam (INN), Oxiracetam [BAN:INN], Oxiracetamum [INN-Latin], CCRIS 4221, Lopac0_000933, O3011_SIGMA, CT-848, CGP 21690E, ISF 2522, ISF-2522, C6H10N2O3, CGP-21690E, 4-Hydroxy-2-oxo-1-pyrrolidineacetamide
InChIKey: IHLAQQPQKRMGSS-UHFFFAOYSA-N | ||||||||
• P-Aminobenzoylanilide
IUPAC Name: N-(4-aminophenyl)benzamide | CAS Registry Number: 17625-83-1 Synonyms: 4'-Aminobenzanilide, P-AMINOBENZALDEHYDE, p-AMINOBENZANILIDE, Benzamide, N-(4-aminophenyl)-, CBMicro_016435, N-(4-Aminophenyl)benzamide, N-Benzoyl-p-phenylenediamine, Oprea1_428735, Oprea1_591737, N-(4-Amino-phenyl)-benzamide, 516090_ALDRICH, ARONIS014451, EINECS 241-603-0, SBB009760, ZINC00123070, BAS 00104927, BIM-0016506.P001, TL8001399, InChI=1/C13H12N2O/c14-11-6-8-12(9-7-11)15-13(16)10-4-2-1-3-5-10/h1-9H,14H2,(H,15,16
InChIKey: GTTFJYUWPUKXJH-UHFFFAOYSA-N | ||||||||
• Palifosfamide
IUPAC Name: bis(2-chloroethylamino)phosphinic acid | CAS Registry Number: 31645-39-3 Synonyms: Ifosfamide mustard, Isophosphamide mustard, Ifosforamide mustard, Isophosphoramide mustard, IPAM, CHEBI:176250, CID100427, NSC297900, NSC 297900, N,N'-Bis(2-chloroethyl)phosphorodiamidic acid, NCI60_002493, Phosphorodiamidic acid, N,N'-bis(2-chloroethyl)-, LS-107954, C16559, N,N'-Di-(2-chloroethyl)phosphorodiamidic acid, N1,N2-Bis(2-chloroethyl)phosphoric acid diamide, 131636-51-6
InChIKey: BKCJZNIZRWYHBN-UHFFFAOYSA-N | ||||||||
• Pamidronic Acid
IUPAC Name: (3-amino-1-hydroxy-1-phosphonopropyl)phosphonic acid | CAS Registry Number: 40391-99-9 Synonyms: pamidronate, Amidronate, Aredia, PAMIDRONIC ACID, Aminomux, AHPrBP, Bisphosphonate 6, pamidronate calcium, pamidronate monosodium, PAMIDRONATE DISODIUM, ChemDiv1_025240, aminopropanehydroxydiphosphonate, Acide pamidronique [INN-French], Acido pamidronico [INN-Spanish], Acidum pamidronicum [INN-Latin], Pamidronic acid [BAN:INN], Pamidronic acid [INN:BAN], C3H11NO7P2, aminohydroxypropylidene diphosphonate, STOCK1N-12562
InChIKey: WRUUGTRCQOWXEG-UHFFFAOYSA-N | ||||||||
• Pelitinib
IUPAC Name: (E)-N-[4-(3-chloro-4-fluoroanilino)-3-cyano-7-ethoxyquinolin-6-yl]-4-(dimethylamino)but-2-enamide | CAS Registry Number: 257933-82-7 Synonyms: EKB-569, Pelitinib (USAN/INN), WAY-EKB 569, WAY-EKB-569, CHEBI:38927, EKB 569, NSC729742, CID6445562, WAY-172569, D05399, (2E)-N-(4-((3-chloro-4-fluorophenyl)amino)-3-cyano-7-ethoxy-6-quinolinyl)-4-(dimethylamino)-2-butenamide, (2E)-N-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamide, (E)-N-[4-(3-Chloro-4-fluoroanilino)-cyano-7-ethoxyquinolin-6-yl]-4-(dimethlyamino)but-2-enamide,, 2-Butenamide, N-(4-((3-chloro-4-fluorophenyl)amino)-3-cyano-7-ethoxy-6-quinolinyl)-4-(dimethylamino)-, (2E)-, 2-Butenamide, N-[4-(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl-4-(dimethylamino)-, (E)-,, 4-Dimethylaminobut-2-enoic Acid, [4-(3-Chloro-4-fluoro phenylamino)-3-cyano-7-ethoxyquinoline-6-yl]amide
InChIKey: WVUNYSQLFKLYNI-AATRIKPKSA-N | ||||||||
• Pelitrexol
IUPAC Name: (2S)-2-[[5-[2-[(6S)-2-amino-4-oxo-5,6,7,8-tetrahydro-1H-pyrido[2,3-d]pyrimidin-6-yl]ethyl]-4-methylthiophene-2-carbonyl]amino]pentanedioic acid | CAS Registry Number: 446022-33-9 Synonyms: Pelitrexol (USAN/INN), UNII-DHT6E8M4KP, AG2037, AG-2032, AG-2037, AG-2038, CID6450821, D05400, (2S)-2-(((5-(2-((6S)-2-Amino-4-oxo-1,4,5,6,7,8-hexahydropyrido(2,3-d)pyrimidin-6-yl)ethyl)-4-methylthiophen-2-yl)carbonyl)amino)pentanedioic acid, L-Glutamic acid, N-((5-(2-((6S)-2-amino-1,4,5,6,7,8-hexahydro-4-oxopyrido(2,3-d)pyrimidin-6-yl)ethyl)-4-methyl-2-thienyl)carbonyl)-
InChIKey: QXOPTIPQEVJERB-JQWIXIFHSA-N | ||||||||
• Perifosine
IUPAC Name: (1,1-dimethylpiperidin-1-ium-4-yl) octadecyl phosphate | CAS Registry Number: 157716-52-4 Synonyms: Perifosine [INN], NKA17, KRX-0401, CID148177, NSC639966, NSC 639966, NSC-639966, D 21266, D-21266, octadecyl-(1,1-dimethyl-4-piperidylio)phosphate, C105905, 4-((Hydroxy(octadecyloxy)phosphinyl)oxy)-1,1-dimethylpiperidinium inner salt, Piperidinium, 4-((hydroxy(octadecyloxy)phosphinyl)oxy)-1,1-dimethyl-, inner salt, Piperidinium, 4-[[hydroxy(octadecyloxy)phosphinyl]oxy]-1,1-dimethyl-, inner salt
InChIKey: SZFPYBIJACMNJV-UHFFFAOYSA-N | ||||||||
• Pharmaceutical Actives | ||||||||
• Pharmaceutical Bulk Active Substances | ||||||||
• Pioglitazone HCL
IUPAC Name: 5-[[4-[2-(5-ethylpyridin-2-yl)ethoxy]phenyl]methyl]-1,3-thiazolidine-2,4-dione hydrochloride | CAS Registry Number: 112529-15-4 Synonyms: Actos, Pioglitazone HCl, Duetact, Glustin, Zactos, Mixture Name, pioglitazone hydrochloride, Actos (TN), C19H20N2O3S.HCl, MLS001306462, MLS001401386, SPECTRUM1504401, Pioglitazone hydrochloride [USAN], U-72107A, CID60560, Pioglitazone hydrochloride (JAN/USP), U-72107E, AD-4833, NCGC00095131-01, NCGC00095131-02
InChIKey: GHUUBYQTCDQWRA-UHFFFAOYSA-N | ||||||||
• Pipendoxifene hydrochloride hydrate
IUPAC Name: 2-(4-hydroxyphenyl)-3-methyl-1-[[4-(2-piperidin-1-ylethoxy)phenyl]methyl]indol-5-ol;hydrate;hydrochloride | CAS Registry Number: 389125-71-7 Synonyms: SCHEMBL6131753, ACM389125717
InChIKey: HDPJXUURTCSOST-UHFFFAOYSA-N | ||||||||
• Pixantrone
IUPAC Name: 6,9-bis(2-aminoethylamino)benzo[g]isoquinoline-5,10-dione | CAS Registry Number: 144510-96-3 Synonyms: 6,9-Aea-biqdo, UNII-F5SXN2KNMR, Pixantrone (USAN/INN), CHEBI:380181, BBR 2778, CID134019, D05522, 6,9-bis(2-aminoethylamino)benzo[g]isoquinoline-5,10-dione, 5,8-Bis((2-aminoethyl)amino)-2-aza-anthracene-9,10-dione, 6,9-Bis((2-aminoethyl)amino)benz(g)isoquinoline-5,10-dione, 6,9-Bis((2-aminoethyl)amino)benzo(g)isoquinoline-5,10-dione, 6,9-Bis-(2-amino-ethylamino)-benzo[g]isoquinoline-5,10-dione, Benz(g)isoquinoline-5,10-dione, 6,9-bis((2-aminoethyl)amino)-
InChIKey: PEZPMAYDXJQYRV-UHFFFAOYSA-N | ||||||||
• Plevitrexed
IUPAC Name: (2S)-2-[[4-[(2,7-dimethyl-4-oxo-1H-quinazolin-6-yl)methyl-prop-2-ynylamino]-2-fluorobenzoyl]amino]-4-(2H-tetrazol-5-yl)butanoic acid | CAS Registry Number: 153537-73-6 Synonyms: Plevitrexed [INN], UNII-L9P2881C3H, ZD 9331, CHEBI:307492, ZD9331, NSC 696259, CID213022, NCI60_034390, LS-184649, (2S)-2-((4-(((2,7-Dimethyl-4-oxo-1,4-dihydroquinazolin-6-yl)methyl)(prop-2-ynyl)amino)-2-fluorobenzoyl)amino)-4-(1H-tetrazol-5-yl)butanoic acid, 1H-Tetrazole-5-butanoic acid, alpha-((4-(((1,4-dihydro-2,7-dimethyl-4-oxo-6-quinazolinyl)methyl)-2-propynylamino)-2-fluorobenzoyl)amino)-, (alphaS)-, 1H-Tetrazole-5-butanoic acid, alpha-((4-(((1,4-dihydro-2,7-dimethyl-4-oxo-6-quinazolinyl)methyl)-2-propynylamino)-2-fluorobenzoyl)amino)-, (S)-, (S)-2-{4-[(2,7-Dimethyl-4-oxo-3,4-dihydro-quinazolin-6-ylmethyl)-prop-2-ynyl-amino]-2-fluoro-benzoylamino}-4-(1H-tetrazol-5-yl)-butyric acid, 172521-94-7
InChIKey: IEJSCSAMMLUINT-NRFANRHFSA-N | ||||||||
• Pomalidomide
IUPAC Name: 4-amino-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione | CAS Registry Number: 19171-19-8 Synonyms: Actimid, 4-Aminothalidomide, IMiD1, IMiD 3, UNII-D2UX06XLB5, IMID-4047, CDC-394, CHEBI:163100, CC-4047, CID134780, CC 4047, 3-Amino-N-(2,6-dioxo-3-piperidyl)phthalimide, Phthalimide, 3-amino-N-(2,6-dioxo-3-piperidyl)-, 4-Amino-2-(2,6-dioxo-3-piperidyl)isoindoline-1,3-dione, 4-amino-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione, 4-Amino-2-(2,6-dioxo-piperidin-3-yl)-isoindole-1,3-dione, 1H-Isoindole-1,3(2H)-dione, 4-amino-2-(2,6-dioxo-3-piperidinyl)-, 443912-23-0, 443919-33-3
InChIKey: UVSMNLNDYGZFPF-UHFFFAOYSA-N | ||||||||
• Pyroxamide
IUPAC Name: N'-hydroxy-N-pyridin-3-yloctanediamide | CAS Registry Number: 382180-17-8 Synonyms: pyroxamide, nchembio.313-comp13, POLAR HYBRID COMPOUND, CID4996, CHEBI:373911, NSC696085, N-Hydroxy-N'-3-pyridinyloctanediamide, NSC-696085, NCI60_034337, Octanediamide, N-hydroxy-N'-3-pyridinyl-, suberoyl-3-aminopyridineamide hydroxamic acid, N-Hydroxy-N'-(3-pyridyl)-1,8-octanediamide, Octanedioic acid hydroxyamide pyridin-3-ylamide
InChIKey: PTJGLFIIZFVFJV-UHFFFAOYSA-N | ||||||||
• Quinagolide
IUPAC Name: (3S,4aS,10aR)-3-(diethylsulfamoylamino)-6-hydroxy-1-propyl-3,4,4a,5,10,10a-hexahydro-2H-benzo[g]quinoline | CAS Registry Number: 87056-78-8 Synonyms: Quinagolide (INN/BAN), CHEBI:157252, CID3086401, D07217, 3-N,N-diethylsulfamide-1-propyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]quinolin-6-ol, (+)N,N-Diethyl-N'-[(3R,4aS,10aS)-1,2,3,4,4a,5,10,10a-octahydro-6-hydroxy-1-proyl-3-benzo[g]quinolinyl]sulfamide, (-)N,N-Diethyl-N'-[(3R,4aS,10aS)-1,2,3,4,4a,5,10,10a-octahydro-6-hydroxy-1-proyl-3-benzo[g]quinolinyl]sulfamide, N,N-Diethyl-N'-[(3R,4aS,10aS)-1,2,3,4,4a,5,10,10a-octahydro-6-hydroxy-1-proyl-3-benzo[g]quinolinyl]sulfamide
InChIKey: GDFGTRDCCWFXTG-ZIFCJYIRSA-N | ||||||||
• Rizatriptan Benzoate
IUPAC Name: benzoic acid; N,N-dimethyl-2-[5-(1,2,4-triazol-1-ylmethyl)-1H-indol-3-yl]ethanamine | CAS Registry Number: 145202-66-0 Synonyms: Maxalt, Rizatriptan benzoate, rizatriptan, Maxalt-MLT, Rizatriptan(RIZ), Maxalt (TN), Rizatriptan Benzoate [USAN], MLS001424197, MK 462, MK-462, MK 0462, MK-0462, Rizatriptan benzoate (JAN/USAN), C15H19N5.C7H6O2, CID77997, CPD000525252, SAM001246615, SMR000525252, L 705126, L-705126
InChIKey: JPRXYLQNJJVCMZ-UHFFFAOYSA-N | ||||||||
• Roquinimex
IUPAC Name: 2-hydroxy-N,1-dimethyl-4-oxo-N-phenylquinoline-3-carboxamide | CAS Registry Number: 84088-42-6 Synonyms: Linomide, ROQUINIMEX, Roquinimexum, Roquinimexum [Latin], Tocris-1461, Quinoline-3-carboxamide, Roquinimex (USAN/INN), Roquinimex [USAN:INN], CCRIS 7673, L1793_SIGMA, LS-2616, FCF 89, FCF-89, PNU-212616, CHEBI:108816, C18H16N2O3, CID55197, LS 2616, NCGC00025172-01, LS-177800
InChIKey: ONCYIVQBAJEKOT-UHFFFAOYSA-N | ||||||||
• Rosabulin
IUPAC Name: 2-[3-[(4-cyanophenyl)methyl]indolizin-1-yl]-N-(3-methyl-1,2-thiazol-5-yl)-2-oxoacetamide | CAS Registry Number: 501948-05-6 Synonyms: Rosabulin (USAN), UNII-6Z674O12T6, CHEBI:535345, STA-5312, CID9843935, D06638, 1-Indolizineacetamide, 3-((4-cyanophenyl)methyl)-N-(3-methyl-5-isothiazolyl)-alpha-oxo-, 2-[3-(4-cyano-benzyl)-3H-indolizin-1-yl]-N-(3-methyl-isothiazol-5-yl)-2-oxo-acetamide, 2-[3-[(4-cyanophenyl)methyl]indolizin-1-yl]-N-(3-methyl-1,2-thiazol-5-yl)-2-oxo-acetamide
InChIKey: IZZYUABKZYIINT-UHFFFAOYSA-N | ||||||||
• Rubitecan
Synonyms: Rubitecan (USAN/INN), D04031
InChIKey: GXSOIDVPIMWEQT-FQEVSTJZSA-N | ||||||||
• Sapacitabine
IUPAC Name: N-[1-[(2R,3S,4S,5R)-3-cyano-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-2-oxopyrimidin-4-yl]hexadecanamide | CAS Registry Number: 151823-14-2 Synonyms: CS-682, CYC-682, CS 682, CID153970, LS-183264, Hexadecanamide, N-(1-(2-cyano-2-deoxy-beta-D-arabinofuranosyl)-1,2-dihydro-2-oxo-4-pyrimidinyl)-, N-(1-(2-cyano-2-deoxy-beta-D-arabinofuranosyl)-1,2-dihydro-2-oxo-4-pyrimidinyl)hexadecanamide
InChIKey: LBGFKUUHOPIEMA-PEARBKPGSA-N | ||||||||
• Semapimod
IUPAC Name: N,N'-bis[3,5-bis[(E)-N-(diaminomethylideneamino)-C-methylcarbonimidoyl]phenyl]decanediamide | CAS Registry Number: 352513-83-8 Synonyms: AXD455, CNI 1493, CNI-1493, AIDS121302, AIDS-121302, CID5745214, N,N'-Bis(3-acetylphenyl)decane diamide tetrakis (amidinohydrazone), N,N'-bis(3,5-bis{(1E)-N-[amino(imino)methyl]ethanehydrazonoyl}phenyl)decanediamide
InChIKey: PWDYHMBTPGXCSN-VCBMUGGBSA-N | ||||||||
• Sodium Valproate
IUPAC Name: sodium 2-propylpentanoate | CAS Registry Number: 1069-66-5 Synonyms: Sodium valproate, Valproate sodium, Depakene, Epilim, Convulex, Eurekene, Labazene, Orfiril, Valerin, Natrium valproat, Selenica, Sodium 2-propylpentanoate, Valproic acid sodium salt, Dipropylacetate sodium, Sodium dipropylacetate, Depakene (TN), Selenica (TN), Sodium bispropylacetate, Valproic acid sodium, Valproinsaeure, natrium
InChIKey: AEQFSUDEHCCHBT-UHFFFAOYSA-M | ||||||||
• Specility Bulk Drug Intermediates | ||||||||
• Sumatriptan Succinate
IUPAC Name: butanedioic acid; 1-[3-(2-dimethylaminoethyl)-1H-indol-5-yl]-N-methylmethanesulfonamide | CAS Registry Number: 103628-48-4 Synonyms: Imigran, Imitrex, Migratriptan, Arcoiran, Micralgin, Migratan, Novelian, Permicran, Sumatrin, Sumigrene, Antibet, Diletan, Imijekt, Sumadol, Migmax, Imigrane, Suminat, SUMATRIPTAN SUCCINATE, Sumavel DosePro, Imitrex (TN)
InChIKey: PORMUFZNYQJOEI-UHFFFAOYSA-N | ||||||||
• Talabostat mesylate
IUPAC Name: [(2S)-1-[(2R)-2-boronopyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]azanium; methanesulfonate | CAS Registry Number: 150080-09-4 Synonyms: Talabostat, Val-boroPro, UNII-V8ZG4Y1B51, Boronic acid, ((2R)-1-((2S)-2-amino-3-methyl-1-oxobutyl)-2-pyrrolidinyl)-, monomethanesulfonate
InChIKey: OXYYOEIGQRXGPI-WSZWBAFRSA-N | ||||||||
• Talampanel
Synonyms: Ampanel, Kinampa, Talampanel (INN), Gyki 53405, GYKI 53773, CHEBI:192577, GYKI-53773, CID164509, IDR-53773, NSC729898, LY 300164, LS-62670, LY-300164, C13670, D02696, (R)-(-)-1-(4-Aminophenyl)-3-acetyl-4-methyl-7,8-methylenedioxy-3,4-dihydro-5H-2,3-benzodiazepine, 7H-1,3-Dioxolo(4,5-h)(2,3)benzodiazepine, 7-acetyl-5-(4-aminophenyl)-8,9-dihydro-8-methyl-, (8R)-, 7H-1,3-Dioxolo(4,5-h)(2,3)benzodiazepine, 7-acetyl-5-(4-aminophenyl)-8,9-dihydro-8-methyl-, (R)-, 7H-1,3-Dioxolo(4,5-h)(2,3)benzodiazepine, 8,9-dihydro-7-acetyl-5-(4-aminophenyl)-8-methyl-, (R)-, 1-[5-(4-Amino-phenyl)-8-methyl-9H-1,3-dioxa-6,7-diaza-cyclohepta[f]inden-7-yl]-ethanone
InChIKey: JACAAXNEHGBPOQ-LLVKDONJSA-N | ||||||||
• Talaporfin sodium
IUPAC Name: tetrasodium (2S)-2-[[2-[(2S,3S)-7-carboxylato-17-ethenyl-12-ethyl-2,8,13,18-tetramethyl-3-(3-oxido-3-oxopropyl)-2,3,23,24-tetrahydroporphyrin-5-yl]acetyl]amino]butanedioate | CAS Registry Number: 220201-34-3 Synonyms: Laserphyrin, Aptocine, Taporfin sodium, Aspartyl chlorin, Monoaspartyl chlorin, NPe6, N-Aspartylchlorin e6, Mono-L-aspartyl chlorin, Mono-L-aspartyl chlorin e6, LS 11 (photosensitizer), LS11, LS 11, LS-11, CID5488036, ME-2906, 220680-62-6, L-Aspartic acid, N-(((7S,8S)-3-carboxy-7-(2-carboxyethyl)-13-ethenyl-18-ethyl-7,8-dihydro-2,8,12,17-tetramethyl-21H,23H-porphin-5-yl)acetyl)-, tetrasodium salt, Tetrasodium (2S)-2-((((7S,8S)-3-carboxylato-7-(2-carboxylatoethyl)-13-ethenyl-18-ethyl-2,8,12,17-tetramethyl-7,8-dihydroporphyrin-5-yl)acetyl)amino)butanedioate
InChIKey: JLWROAPZCOJYGT-OBJGRMLXSA-J | ||||||||
• Taltobulin
IUPAC Name: (E,4S)-4-[[(2S)-3,3-dimethyl-2-[[(2S)-3-methyl-2-(methylamino)-3-phenylbutanoyl]amino]butanoyl]-methylamino]-2,5-dimethylhex-2-enoic acid | CAS Registry Number: 228266-40-8 Synonyms: Taltobulin (USAN/INN), HTI-286, SPA-110, CHEBI:406312, CID6918637, D06001, (E)-(S)-4-{[(S)-3,3-Dimethyl-2-((S)-3-methyl-2-methylamino-3-phenyl-butyrylamino)-butyryl]-methyl-amino}-2,5-dimethyl-hex-2-enoic acid, (S)-2,5-dimethyl-4-((S)-N,3,3-trimethyl-2-((S)-3-methyl-2-(methylamino)-3-phenylbutanamido)butanamido)hex-2-enoic acid, (S,E)-2,5-dimethyl-4-((S)-N,3,3-trimethyl-2-((S)-3-methyl-2-(methylamino)-3-phenylbutanamido)butanamido)hex-2-enoic acid, 4-{[3,3-Dimethyl-2-(3-methyl-2-methylamino-3-phenyl-butyrylamino)-butyryl]-methyl-amino}-2,5-dimethyl-hex-2-enoic acid, N,beta,beta-trimethyl-L-phenylalanyl-N-[(3S,4E)-5-carboxy-2-methylhex-4-en-3-yl]-N,3-dimethyl-L-valinamide
InChIKey: CNTMOLDWXSVYKD-PSRNMDMQSA-N | ||||||||
• Tamibarotene
IUPAC Name: 4-[(5,5,8,8-tetramethyl-6,7-dihydronaphthalen-2-yl)carbamoyl]benzoic acid | CAS Registry Number: 94497-51-5 Synonyms: Amnoid, Amnolake, Amnoleuk, Tamibaro, retinobenzoic acid, 2cbr, Am 80, Amnoid (TN), Am80, Tamibarotene (JAN/INN), UNII-08V52GZ3H9, AM-80, TOS-80, CHEBI:32181, NSC608000, AIDS130644, NSC 608000, AIDS-130644, CID108143, TM-411
InChIKey: MUTNCGKQJGXKEM-UHFFFAOYSA-N | ||||||||
• Tariquidar
IUPAC Name: N-[2-[[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]-4,5-dimethoxyphenyl]quinoline-3-carboxamide | CAS Registry Number: 206873-63-4 Synonyms: tariquidarth, Tariquidar (USAN/INN), UNII-J58862DTVD, CHEBI:359664, XR9576, XR 9576, CID148201, D06008, C402343, N-(2-((4-(2-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)ethyl)phenyl)carbamoyl)-4,5-dimethoxyphenyl)quinoline-3-carboxamide, 1N-{4-[2-(6,7-dimethoxy-1,2,3,4-tetrahydro-2-isoquinolinyl)ethyl]phenyl}-4,5-dimethoxy-2-(3-quinolylcarboxamido)benzamide, 3-Quinolinecarboxamide, N-(2-(((4-(2-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)ethyl)phenyl)amino)carbonyl)-4,5-dimethoxyphenyl)-
InChIKey: LGGHDPFKSSRQNS-UHFFFAOYSA-N | ||||||||
• Tasidotin hydrochloride
IUPAC Name: (2S)-N-tert-butyl-1-[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-(dimethylamino)-3-methylbutanoyl]amino]-3-methylbutanoyl]-methylamino]-3-methylbutanoyl]pyrrolidine-2-carbonyl]pyrrolidine-2-carboxamide hydrochloride | CAS Registry Number: 623174-20-9 Synonyms: Tasidotin HCl, Tasidotin hydrochloride (USAN), ILX 651, BSF 223651, CID11479259, LU 223651, D06009, 848866-34-2
InChIKey: OOKIODJYZSVHDO-QMYFOHRPSA-N | ||||||||
• Terameprocol
IUPAC Name: 4-[4-(3,4-dimethoxyphenyl)-2,3-dimethylbutyl]-1,2-dimethoxybenzene | CAS Registry Number: 5701-82-6 Synonyms: Tmndga, Tetra-O-methyl-ndga, Dimethyldihydroguaiaretic acid, NORDIHYDROGUAIARETIC ACID, Tetramethoxynordihydroguaiaretic acid, tetra-O-methyl nordihydroguaiaretic acid, CHEBI:562175, NSC 136955, Tetra-O-methylnordihydroguaiaretic acid, CID97616, NSC136955, FW 358.2, LS-29888, meso-1,4-Bis(3,4-dimethoxyphenyl)dimethylbutane, 1,4-Bis(3,4-dimethoxyphentl)-2,3-dimethylbutane, 4,4'-(2,3-Dimethyl-1,4-butanediyl)bis-1,2-dimethoxybenzene, Butane, 1,4-bis(3,4-dimethoxyphenyl)-2,3-dimethyl-, 1,1'-(2,3-Dimethyl-1,4-butanediyl)bis(3,4-dimethoxybenzene), Benzene, 1,1'-(2,3-dimethyl-1,4-butanediyl)bis(3,4-dimethoxy-, Benzene, 1,1'-(2,3-dimethyl-1,4-butanediyl)bis[3,4-dimethoxy]
InChIKey: ORQFDHFZSMXRLM-UHFFFAOYSA-N | ||||||||
• Tesmilifene
IUPAC Name: 2-(4-benzylphenoxy)-N,N-diethylethanamine | CAS Registry Number: 98774-23-3 Synonyms: Depmpe, DPPE hydrochloride, Tocris-0743, UNII-I43T3ID6G2, C19H25NO, CHEBI:135953, 92981-78-7 (hydrochloride), CID108092, NCGC00024762-01, NCGC00024762-02, 2-((alpha-Phenyl-p-tolyl)oxy)triethylamine, LS-178389, [2-(4-Benzyl-phenoxy)-ethyl]-diethyl-amine, N,N-Diethyl-2-((4-phenylmethyl)phenoxy)ethanamine, Ethanamine, N,N-diethyl-2-(4-(phenylmethyl)phenoxy)-, N,N-diethyl-2-(4-(phenylmethyl)phenoxy)ethanamine, BRD-K80315159-051-01-2, N,N-diethyl-2-(4-(phenylmethyl)phenoxy)ethanamine hydrochloride, Ethanamine, N,N-diethyl-2-(4-(phenylmethyl)phenoxy)-, (2aR-(2aalpha,4beta,4abeta,6beta,9alpha(alphaR*,betaS*),11alpha,12alpha,12aalpha,12balpha))-
InChIKey: NFIXBCVWIPOYCD-UHFFFAOYSA-N | ||||||||
• Tipifarnib
IUPAC Name: 6-[(R)-amino-(4-chlorophenyl)-(3-methylimidazol-4-yl)methyl]-4-(3-chlorophenyl)-1-methylquinolin-2-one | CAS Registry Number: 192185-72-1 Synonyms: Zarnestra, Tipifarnib [USAN], Tipifarnib (USAN/INN), 1x81, CID159324, NSC-702818, LS-184411, LS-187005, LS-187640, (R)-( )-R115777, D03720, R115777, (R)-( )-R-115777, R-115777, (R)-6-(Amino(4-chlorophenyl)(1-methyl-1H-imidazol-5-yl)methyl)-4-(3-chlorophenyl)-1-methyl-2(1H)-quinolinone, 2 (1H))-Quinolinone,6-(amino(4-chlorophenyl)(1-methyl-1H-imidazol-5-yl)methyl)-4-(3-chlorophenyl)-1-methyl-, 2(1H )-quinolinone, JAN, 2 (1H))-Quinolinone,6-(amino(4-chlorophenyl)(1-methyl-1H-imidazol-5-yl)methyl)-4-(3-chlorophenyl)-1-methyl-, (+)-, 6-[(R)-amino(4-chlorophenyl)(1-methyl-1H-imidazol-5-yl)methyl]-4-(3-chlorophenyl)-1-methylquinolin-2(1H)-one, 6-[(S)-AMINO(4-CHLOROPHENYL)(1-METHYL-1H-IMIDAZOL-5-YL)METHYL]-4-(3-CHLOROPHENYL)-1-METHYLQUINOLIN-2(1H)-ONE
InChIKey: PLHJCIYEEKOWNM-HHHXNRCGSA-N | ||||||||
• Triciribine
Synonyms: Tricyclic nucleoside, Pentaazacentopthylene, API-2, Akt Inhibitor V, Triciribine, NSC154020, Akt/PKB Signaling Inhibitor-2, CID290486, HSCI1_000386, NCGC00014417, NSC 154020, NCI60_001091, BRD-A42649439-001-01-0, TCN, 1,4,5,6,8-Pentaazaacenaphthylene, 3-amino-1,5-dihydro-5-methyl-1-.beta.-D-ribofuranosyl, 1,4,5,6,8-Pentaazaacenaphthylene, 3-amino-1,5-dihydro-5-methyl-1-.beta.-D-ribofuranosyl-, 1,4,5,6,8-Pentaazaacennaphthylen-3-amine, 1,5-dihydro-5-methyl-1-.beta.-D-ribofuranosyl-
InChIKey: HOGVTUZUJGHKPL-UHFFFAOYSA-N | ||||||||
• Troxacitabine
IUPAC Name: 4-amino-1-[(2S,4S)-2-(hydroxymethyl)-1,3-dioxolan-4-yl]pyrimidin-2-one | CAS Registry Number: 145918-75-8 Synonyms: cis-Dioxolane-C, L-1,3-dioxolane-cytidine, (-)-L-.b.-DioxolaneC, Troxacitabine (USAN/INN), CHEBI:349301, AIDS004371, (-)-L-.beta.-Dioxolane-cytosine, AIDS-004371, CID454194, NSC668281, ZINC01642845, D06255, (-)-(2S,4S)-1-[2-Hydroxymethyl)-1,3-dioxolan-4-yl]cytosine, 4-Amino-1-(2-hydroxymethyl-[1,3]dioxolan-4-yl)-1H-pyrimidin-2-one, LTT
InChIKey: RXRGZNYSEHTMHC-BQBZGAKWSA-N | ||||||||
• Vandetanib
IUPAC Name: N-(4-bromo-2-fluorophenyl)-6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-amine | CAS Registry Number: 338992-00-0 Synonyms: Zactima, vande-tanib, Vandetanib [INN], 2ivu, Vandetanib (JAN/INN), ZD6474, CHEBI:49960, ZD 6474, ZD-6474, AZD-6474, CID3081361, NCGC00167513-01, LS-184394, D06407, C452423, N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-((1-methyl-4-piperidinyl)methoxy)-4-quinazolinamine, N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-((1-methylpiperidin-4-yl)methoxy)quinazolin-4-amine, 4-Quninazolinamine, N-(4-bromo-2-fluorophenyl)-6-methoxy-7-((1-methyl-4-piperidinyl)methoxy)-, 443913-73-3, N-(4-bromo-2-fluorophenyl)-6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-amine
InChIKey: UHTHHESEBZOYNR-UHFFFAOYSA-N | ||||||||
• Vatalanib Succinate
IUPAC Name: butanedioic acid; N-(4-chlorophenyl)-4-(pyridin-4-ylmethyl)phthalazin-1-amine | CAS Registry Number: 212142-18-2 Synonyms: Vatalanib succinate, PTK/ZK, Ptk 787, PTK-787, PTK787, CGP 79787D, CGP-79787D, CGP-79787, ZK 222584, LS-186035, ZK-222584, 1-Phthalazinamine, N-(4-chlorophenyl)-4-(4-pyridinylmethyl)-, butanedioate (1:1), Butanedioic acid, compd. with N-(4-chlorophenyl)-4-(4-pyridinylmethyl)-1-phthalazinamine (1:1)
InChIKey: LLDWLPRYLVPDTG-UHFFFAOYSA-N | ||||||||
• Verteporfin
Synonyms: Visudyne, Visudyne (TN), VERTEPORFIN, Verteporfin (JAN/USAN/INN), NCGC00017148-01, CAS-129497-78-5, D01162
InChIKey: NJLRKAMQPVVOIU-IDLGWYNRSA-N | ||||||||
• Xaliproden hydrochloride
IUPAC Name: 1-(2-naphthalen-2-ylethyl)-4-[3-(trifluoromethyl)phenyl]-3,6-dihydro-2H-pyridine hydrochloride | CAS Registry Number: 90494-79-4 Synonyms: Xaprila, SR 57746A, SR-57746A, Xaliproden hydrochloride (JAN), MolPort-003-666-826, CID128918, SR-57746, LS-132040, D01537, 1-(2-(Naphth-2-yl)ethyl)-4-(3-trifluoromethylphenyl)-1,2,5,6-tetrahydropyridine hydrochloride, Pyridine, 1,2,3,6-tetrahydro-1-(2-(2-naphthalenyl)ethyl)-4-(3-(trifluoromethyl)phenyl)-, hydrochloride
InChIKey: WVHBEIJGAINUBW-UHFFFAOYSA-N | ||||||||
• Zaleplon
IUPAC Name: N-[3-(3-cyanopyrazolo[1,5-a]pyrimidin-7-yl)phenyl]-N-ethylacetamide | CAS Registry Number: 151319-34-5 Synonyms: zaleplon, Sonata, Zerene, Sonata (TN), Zaleplon [USAN:INN], DEA No. 2781, Zaleplon (JAN/USAN/INN), MLS000759451, ZAL 846, C17H15N5O, LJC 10846, BB_SC-4140, SKP-1041, AZ-007, LJC-10846, L846, CL-284846, DB00962, LS-8737, CL 284,846
InChIKey: HUNXMJYCHXQEGX-UHFFFAOYSA-N | ||||||||
• Ziprasidone
IUPAC Name: 5-[2-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]ethyl]-6-chloro-1,3-dihydroindol-2-one | CAS Registry Number: 146939-27-7 Synonyms: Zeldox, ziprazidone, Geodon, Ambap6301, Ziprasidone hydrochloride, Ziprasidone [INN:BAN], C21H21ClN4OS, MLS000759435, Ziprasidone mesylate trihydrate, CHEBI:10119, CID60854, DB00246, CP 88059, CPD000466328, LS-83744, SAM001246607, SMR000466328, CP-88,059, TL8000889, CP 88059-01
InChIKey: MVWVFYHBGMAFLY-UHFFFAOYSA-N | ||||||||
• Zolmitriptan
IUPAC Name: (4S)-4-[[3-(2-dimethylaminoethyl)-1H-indol-5-yl]methyl]-1,3-oxazolidin-2-one | CAS Registry Number: 139264-17-8 Synonyms: zolmitriptan, Zomig, Zomigon, Flezol, AscoTop, Zomig Nasal Spray, Zomig ZMT, Zomig-ZMT, Zolmitriptan [USAN], Spectrum2_000728, MLS000758208, MLS001424172, SPECTRUM1505281, SPBio_000656, CHEBI:10124, C16H21N3O2, CID60857, 311C90, BW-311C90, CPD000449310
InChIKey: ULSDMUVEXKOYBU-ZDUSSCGKSA-N | ||||||||
• Zolpidem
IUPAC Name: N,N-dimethyl-2-[6-methyl-2-(4-methylphenyl)imidazo[1,2-a]pyridin-3-yl]acetamide | CAS Registry Number: 82626-48-0 Synonyms: zolpidem, Lorex, Ambien, Zolpidemum [Latin], ZOLPIDEM TARTRATE, Zolpidem [INN:BAN], Z103_SIGMA, DEA No. 2783, BSPBio_002278, SPECTRUM1505369, STOCK6S-53875, CID5732, 2C19H21N3O, DB00425, SL-800750, NCGC00095179-01, NCGC00095179-02, NCGC00095179-03, NCGC00095179-04, LS-80196
InChIKey: ZAFYATHCZYHLPB-UHFFFAOYSA-N | ||||||||
• Zosuquidar
Synonyms: NCGC00274062-01, Zosuquidar Hydrochloride, AC1MI1NN, 167465-36-3, SureCN12432743, CHEMBL444172, CS-0921, RL02146, HY-15255, RS 33295-198, Zosuquidar|167354-41-8|LY 335979|LY-335979, (|AR)-4-[(1a|A,6|A,10b|A)-1,1-Difluoro-1,1a,6,10b-tetrahydrodibenzo[a,e]cyclopropa[c]cyclohepten-6-yl]-|A-[(5-quinolinyloxy)methyl]-1-piperazineethanol Hydrochloride, (2R)-1-{4-[(1aR,6r,10bS)-1,1-Difluoro-1,1a,6,10b-tetrahydrodibenzo[a,e]cyclopropa[c]cyclohepten-6-yl]piperazin-1-yl}-3-(quinolin-5-yloxy)propan-2-ol
InChIKey: IHOVFYSQUDPMCN-XAKVHENESA-N | ||||||||
• 1-Methoxyl-2-Adamantyl-4-Bromo-Benzene | ||||||||
• 3-Aminopyridine-2-carboxaldehyde-thiosemicarbazone
IUPAC Name: [(E)-(3-aminopyridin-2-yl)methylideneamino]thiourea | CAS Registry Number: 236392-56-6 Synonyms: Triapine, 3-Apct, Pan 811, 3-AP, C7H9N5S, OCX 191, CHEBI:483750, AIDS179996, NSC 663249, AIDS-179996, NSC663249, CID9571836, 3-Aminopyridine-2-carboxaldehyde thiosemicarbazone, LS-76467, 3-Aminopyridine-2-carboxaldehyde- thiosemicarbazone, 3-aminopyridine-2-carbaldehyde thiosemicarbazone, 1-((3-aminopyridin-2-yl)methylene)thiosemicarbazide, Hydrazinecarbothioamide, 2-((3-amino-2-pyridinyl)methylene)-, -AP, 143621-35-6
InChIKey: XMYKNCNAZKMVQN-NYYWCZLTSA-N |