Profile: Jinan Trio PharmaTech Co., Ltd. specializes in APIs & intermediates, heterocyclic compounds, and anti-tumor drugs. Our products include crizotinib, vemurafenib, afatinib, vandetanib, regorafenib, brivanib alaninate, pyridazine, imidazole, pyrazole, and oxazole. We are specialized in providing over 1000 products including molecular targeted anticancer drugs, cell signaling pathway inhibitors, pharmaceutical intermediates, and heterocyclic compounds, and quality services including custom synthesis, transfer of new drug patent and technology, technical cooperation, and process optimization.
• ETHYL 4-NITRO-1H-IMIDAZOLE-2-CARBOXYLATE
IUPAC Name: ethyl 5-nitro-1H-imidazole-2-carboxylate | CAS Registry Number: 865998-46-5 Synonyms: Ethyl 5-nitro-1H-imidazole-2-carboxylate, ethyl 4-nitro-1H-imidazole-2-carboxylate, 4-NITRO-1H-IMIDAZOLE-2-CARBOXYLIC ACID ETHYL ESTER, PubChem23761, SureCN1595448, CTK5F6999, ANW-44975, AKOS006285014, AKOS015901682, AB44510, ACN-000290, AG-H-49317, AK-80184, KB-65173, 1H-Imidazole-2-carboxylic acid,5-nitro-,ethyl ester, 1H-Imidazole-2-carboxylicacid, 5-nitro-, ethyl ester, I14-14335, 1H-Imidazole-2-carboxylicacid, 4-nitro-, ethyl ester (9CI);4-Nitro-1H-imidazole-2-carboxylic acid ethylester;Ethyl 5-nitro-1H-imidazole-2-carboxylate;
InChIKey: YSVPLWXCZZORIO-UHFFFAOYSA-N | ||||||||
• ethyl 5-amino-6-bromo-2-methylnicotinate
IUPAC Name: ethyl 5-amino-6-bromo-2-methylpyridine-3-carboxylate | CAS Registry Number: 1149388-64-6 Synonyms: Ethyl 5-amino-6-bromo-2-methylnicotinate, AKOS016011825, AK123504, KB-253586
InChIKey: AAMKCVXAHVFSND-UHFFFAOYSA-N | ||||||||
• Ethyl 5-formyl-2,4-dimethyl-1H-pyrrole-3-carboxylate
IUPAC Name: ethyl 5-formyl-2,4-dimethyl-1H-pyrrole-3-carboxylate | CAS Registry Number: 2199-59-9 Synonyms: NSC13426, ZINC01729614, SL-00002, 5-Formyl-2,4-dimethyl-1H-pyrrole-3-carboxylic acid ethyl ester, 1H-Pyrrole-3-carboxylic acid, 5-formyl-2,4-dimethyl-, ethyl ester
InChIKey: GDISALBEIGGPER-UHFFFAOYSA-N | ||||||||
• Ethyl 6-methylimidazo[2,1-b]thiazole-5-carboxylate
IUPAC Name: ethyl 6-methylimidazo[2,1-b][1,3]thiazole-5-carboxylate | CAS Registry Number: 57626-37-6 Synonyms: ethyl 6-methylimidazo[2,1-b][1,3]thiazole-5-carboxylate, ethyl 3-methyl-imidazo[2,1-b]thiazole 4-carboxylate, AG-G-03517, ST019484, BAS 00602579, AC1LDOF3, CBMicro_025689, ChemDiv2_003962, SureCN952278, AC1Q32ML, KSC607C8P, MLS000061584, CTK5A7187, MolPort-000-423-264, HMS1380E02, HMS2459N13, ANW-48821, CCG-12662, ZINC00032013, AKOS000118207
InChIKey: NSUFDDBQLKSSIN-UHFFFAOYSA-N | ||||||||
• ethyl imidazo[2,1-b]thiazole-5-carboxylate
IUPAC Name: ethyl imidazo[2,1-b][1,3]thiazole-5-carboxylate | CAS Registry Number: 349480-83-7 Synonyms: Ethyl imidazo[2,1-b]thiazole-5-carboxylate, SureCN1338053, CTK8C2940, ANW-69334, RW4013, AKOS016005785, AK-31310, QC-10487, KB-134791
InChIKey: YVUGUFMTQJLGPE-UHFFFAOYSA-N | ||||||||
• Ethyl Imidazole-2-Carboxylate
IUPAC Name: ethyl 1H-imidazole-2-carboxylate | CAS Registry Number: 33543-78-1 Synonyms: Ethyl 1H-imidazole-2-carboxylate, Imidazole, 2-ethoxycarbonyl-, Ethyl imidazole-2-carboxylate, CID549404, OR3003, TE6113, ZINC12360040
InChIKey: UHYNYIGCGVDBTC-UHFFFAOYSA-N | ||||||||
• Ethyl isocyanoacetate
IUPAC Name: ethyl 2-isocyanoacetate | CAS Registry Number: 2999-46-4 Synonyms: 226319_ALDRICH, 58822_FLUKA, EINECS 221-077-9, InChI=1/C5H7NO2/c1-3-8-5(7)4-6-2/h3-4H2,1H
InChIKey: FPULFENIJDPZBX-UHFFFAOYSA-N | ||||||||
• Ethyl oxazole-2-carboxylate
IUPAC Name: ethyl 1,3-oxazole-2-carboxylate | CAS Registry Number: 33036-67-8 Synonyms: ETHYL OXAZOLE-2-CARBOXYLATE, Ethyl 2-oxazolecarboxylate, ethyl 1,3-oxazole-2-carboxylate, Oxazole-2-carboxylic acid ethyl ester, 2-OXAZOLECARBOXYLIC ACID, ETHYL ESTER, PubChem15936, ACMC-209hy0, AGN-PC-01WF5R, SureCN2422303, CTK4G9792, MolPort-004-780-531, ACN-S001772, 2-Oxazolecarboxylicacid, ethyl ester, ANW-27526, WTI-10524, AKOS006280725, AB19317, AG-F-10956, RP20661, AK-68691
InChIKey: JYQRCIRWXOYCLA-UHFFFAOYSA-N | ||||||||
• Ethyl-4-hydroxy-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxylate
IUPAC Name: (3Z)-3-[ethoxy(hydroxy)methylidene]-6-methyl-1H-pyridine-2,4-dione | CAS Registry Number: 10350-10-4 Synonyms: Maybridge3_000642, Oprea1_491016, MLS000736242, MLS000737690, TPC-PY051, BTB 12129, NSC109231, Ethyl 2,4-dihydroxy-6-methylnicotinate, IDI1_012029, 11L-585S, SMR000338492, 3-Pyridinecarboxylic acid, 1,2-dihydro-4-hydroxy-6-methyl-2-oxo-, ethyl ester, ethyl 4-hydroxy-6-methyl-2-oxo-1,2-dihydro-3-pyridinecarboxylate, Ethyl Ester, 2,4-Dihydroxy-6-Methyl-3-Pyridine Carboxylic Acid, 70254-52-3
InChIKey: YSUHDCOUISXHEX-CLFYSBASSA-N | ||||||||
• Ethyl1-methyl-4-nitroimidazole-2-carboxylate
IUPAC Name: ethyl 1-methyl-4-nitroimidazole-2-carboxylate | CAS Registry Number: 109012-23-9 Synonyms: ethyl 1-methyl-4-nitroimidazole-2-carboxylate, ethyl 1-methyl-4-nitro-1H-imidazole-2-carboxylate, ethyl 4-nitro-1-methylimidazole-2-carboxylate, Ethyl-1-methyl-4-nitroimidazole-2-carboxylate, 1H-Imidazole-2-carboxylicacid, 1-methyl-4-nitro-, ethyl ester, ZINC02511034, PubChem23738, AC1MBZ4Q, ACMC-1BSR3, SureCN1594419, CTK4A6291, MolPort-000-155-301, ACN-P000771, ANW-50541, SBB092420, AKOS006277851, AB16105, AG-D-25730, RP25681, AK-22184
InChIKey: QGTGFMLXIBQONB-UHFFFAOYSA-N | ||||||||
• Ethyl2,5-dibroMooxazole-4-carboxylate
IUPAC Name: ethyl 2,5-dibromo-1,3-oxazole-4-carboxylate | CAS Registry Number: 862731-70-2 Synonyms: Ethyl 2,5-dibromooxazole-4-carboxylate, ZINC32602816, AKOS015951462, KB-77260, AB1010135, X0320, 460081-22-5
InChIKey: FJGMBUMDLBUTNO-UHFFFAOYSA-N | ||||||||
• Everolimus
Synonyms: Certican, Afinitor, Everolimus [USAN], SDZ-RAD, RAD001, NVP-RAD-001, RAD 001, RAD-001C, 42-O-(2-Hydroxyethyl)rapamycin, RAD-001, Rapamycin, 42-O-(2-hydroxyethyl)-, 42-O-(2-Hydroxy)ethyl rapamycin, NCGC00167512-01, LS-143292, (1R,9S,12S,15R,16E,18R,19R,21R,23S,24E,26E,28E,30S,32S,35R)-1,18-Dihydroxy-12-((1R)-2-((1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl)-1-methylethyl)-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo(30.3.1.04,9)hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentaone, RAD, (1R,9S,12S,15R,16E,18R,19R,21R,23S,24E,26E,28E,30S,32S,35R)-1,18-Dihydroxy-12-((1R)-2-((1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl)-1-methylethyl)-19,30-dimethoxy-15,17,21,23,29,35-hexamethyl-11,36-dioxa-4-azatricyclo(30.3.1.0(sup 4,9))hexatriaconta-16,24,26,28-tetraene-2,3,10,14,20-pentaone, (3S,6R,7E,9R,10R,12R,14S,15E,17E,19E,21S,23S,26R,27R,34aS)-9,10,12,13,14,21,22,23,24,25,26,27,32,33,34,34a-Hexadecahydro-9,27-dihydroxy-3-((1R)-2-((1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl)-1-methylethyl)-10,21-dimethoxy-6,8,12,14,20,26-hexamethyl-23,27-epoxy-3H-pyrido(2,1-c)(1,4)oxaazacyclohentriacontine-1,5,11,28,29(4H,6H,31H)-pentone, (3S,6R,7E,9R,10R,12R,14S,15E,17E,19E,21S,23S,26R,27R,34aS)-9,27-dihydroxy-3-{(2R)-1-[(1S,3R,4R)-4-(2-hydroxyethoxy)-3-methoxycyclohexyl]propan-2-yl}-10,21-dimethoxy-6,8,12,14,20,26-hexamethyl-9,10,12,13,14,21,22,23,24,25,26,27,32,33,34,34a-hexadecahydro-3H-23,27-epoxypyrido[2,1-c][1,4]oxazacyclohentriacontine-1,5,11,28,29(4H,6H,31H)-pentone
InChIKey: HKVAMNSJSFKALM-GKUWKFKPSA-N | ||||||||
• Fasudil Hydrochloride
IUPAC Name: 5-(1,4-diazepan-1-ylsulfonyl)isoquinoline hydrochloride | CAS Registry Number: 105628-07-7 Synonyms: Fasudil hydrochloride, Fasudil, Fasdil, Eril, AT 877 hydrochloride, HA 1077 hydrochloride, Fasudil hydrochloride (JAN), C14H17N3O2S.HCl, MLS000069344, ha-1077, HA-1077 DIHYDROCHLORIDE, AT-877, CID163751, NCGC00180915-01, LS-60222, SMR000058993, D01840, 1H-1,4-Diazepine, hexahydro-1-(5-isoquinolinylsulfonyl)-, monohydrochloride, Hexahydro-1-(5-isoquinolinylsulfonyl)-1H-1,4-diazepine monohydrochloride, 133337-43-6
InChIKey: LFVPBERIVUNMGV-UHFFFAOYSA-N | ||||||||
• Flavopiridol
IUPAC Name: 2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3R,4S)-3-hydroxy-1-methylpiperidin-4-yl]chromen-4-one | CAS Registry Number: 146426-40-6 Synonyms: nchembio.90-comp9, CID5459219, NCI60_017396, L 868275, L-868275, L86-8275, (-)-2-(2-Chlorophenyl)-5,7-dihydroxy-8-[(3R,4S)-3-hydroxy-1-methyl-4-piperidinyl]-4H-1-benzopyran-4-one, (-)cis-5,7-Dihydroxy-2-(2-chlorophenyl)-8-(4-(3-hydroxy-1-methyl)piperidinyl)-4H-1-benzopyran-4-one, 4H-1-Benzopyran-4-one, 2-(2-chlorophenyl)-5,7-dihydroxy-8-((3R,4S)-3-hydroxy-1-methyl-4-piperidinyl)-, rel-(-)-, 4H-1-Benzopyran-4-one, 2-(2-chlorophenyl)-5,7-dihydroxy-8-(3-hydroxy-1-methyl-4-piperidinyl)-, cis-(-)-
InChIKey: BIIVYFLTOXDAOV-PXAZEXFGSA-N | ||||||||
• Flavopiridol hydrochloride
IUPAC Name: 2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]chromen-4-one hydrochloride | CAS Registry Number: 131740-09-5 Synonyms: Alvocidib, Alvocidib (USAN/INN), F3055_SIGMA, NSC-649890, D02880, L-86-8276, (-)-2-(2-Chlorophenyl)-5,7-dihydroxy-8-[(3s,4r)-3-hydroxy-1-methyl-4-piperidinyl]-4h-1-benzopyran-4-one hydrochloride
InChIKey: LGMSNQNWOCSPIK-LWHGMNCYSA-N | ||||||||
• Fludarabine
IUPAC Name: [(2R,3S,4S,5R)-5-(6-amino-2-fluoropurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl dihydrogen phosphate | CAS Registry Number: 75607-67-9 Synonyms: fludara, fludarabine phosphate, Fludura, Beneflur, FAMP, FaraAMP, fluoro-ara-AMP, Fludarabine monophosphate, 2-Fluoro-ARA AMP, Fludara (TN), 2-Fluoro-ara-AMP, F-ara-AMP, Ambap1079, Fludarabine 5'-monophosphate, 2-F-ara-AMP, C10H13FN5O7P, Fludarabine phosphate [USAN:BAN], NSC-312887, Fludarabine phosphate (JAN/USP), SHT-586
InChIKey: GIUYCYHIANZCFB-FJFJXFQQSA-N | ||||||||
• Fludarabine (base)
IUPAC Name: (2R,3S,4S,5R)-2-(6-amino-2-fluoropurin-9-yl)-5-(hydroxymethyl)oxolane-3,4-diol | CAS Registry Number: 21679-14-1 Synonyms: Fludarabine, fludara, FaraA, SQ Fludarabine, 2-Fluoro Ara-A, Fludarabinum [Latin], Fludarabina [Spanish], F-Ara-A, Fludarabine [INN], fludarabine phosphate, 2-F-ara-A, CCRIS 3382, HSDB 6964, MLS000028687, C10H12FN5O4, EINECS 244-525-5, NSC 118218H, NSC 118218, 9-beta-D-Arabinosyl-2-fluoroadenine, 2-Fluoro-9-beta-D-arabinofuranosyladenine
InChIKey: HBUBKKRHXORPQB-FJFJXFQQSA-N | ||||||||
• FMK
IUPAC Name: 1-[4-amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)pyrrolo[2,3-d]pyrimidin-6-yl]-2-fluoroethanone | CAS Registry Number: 821794-92-7 Synonyms: AC1LD8U9, CHEMBL515414, CHEBI:558490, HY-52101A, CS-0648, QC-8903, KB-77351, fluoromethylketone-pyrrolopyrimidine scaffold, FMK|821794-92-7, S7064,1111636-35-1, 1-(4-amino-7-(3-hydroxypropyl)-5-p-tolyl-7H-pyrrolo[2,3-d]pyrimidin-6-yl)-2-fluoroethanone, 1-[4-Amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]-2-fluoroethanone, 1-[4-amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)pyrrolo[2,3-d]pyrimidin-6-yl]-2-fluoroethanone, ethanone, 1-[4-amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]-2-fluoro-, Ethanone, 1-[4-amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]-2-fluoro- (9CI)
InChIKey: IKLGYJACVCXYIL-UHFFFAOYSA-N | ||||||||
• FORMAMIDE,N-1H-BENZO[D]IMIDAZOL-4-YL-
IUPAC Name: N-(1H-benzimidazol-4-yl)formamide | CAS Registry Number: 137654-47-8 Synonyms: N-(1H-Benzo[d]imidazol-4-yl)formamide, CTK8C2323, MolPort-004-752-554, ANW-68204, AKOS016007144, AK-80616
InChIKey: LGITZGIQYPDWBF-UHFFFAOYSA-N | ||||||||
• Fostamatinib Disodium
IUPAC Name: [6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)pyrimidin-4-yl]amino]-2,2-dimethyl-3-oxopyrido[3,2-b][1,4]oxazin-4-yl]methyl dihydrogen phosphate | CAS Registry Number: 901119-35-5 Synonyms: Fostamatinib, R788, Fostamatinib, R7935788, R 788, 2H-Pyrido(3,2-b)-1,4-oxazin-3(4H)-one, 6-((5-fluoro-2-((3,4,5-trimethoxyphenyl)amino)-4-pyrimidinyl)amino)-2,2-dimethyl-4-((phosphonooxy)methyl)-, 2H-Pyrido[3,2-b]-1,4-oxazin-3(4H)-one, 6-[[5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]-4-pyrimidinyl]amino]-2,2-dimethyl-4-[(phosphonooxy)methyl]-, R788 compound, Fostamatinib (USAN), S2625_Selleck, R-788 Free acid, R788 (Fostamatinib), AGN-PC-00DTWF, Fostamatinib [USAN:INN], R788 FREE ACID, R-935788 Free acid, SureCN1201371, UNII-SQ8A3S5101, QCR-82, CHEMBL2103830, R935788 FREE ACID
InChIKey: GKDRMWXFWHEQQT-UHFFFAOYSA-N | ||||||||
• FURO[2,3-C]PYRIDIN-3(2H)-ONE
IUPAC Name: furo[2,3-c]pyridin-3-one | CAS Registry Number: 106531-52-6 Synonyms: AG-D-21014, PubChem24154, ACMC-20c3nr, SureCN4822863, AGN-PC-000OO8, Furo[2,3-c]pyridin-3-one;, CTK0H2643, MolPort-004-757-821, RW3067, AKOS016011729, QC-1965, AK123377, Furo[2,3-c]pyridin-3(2H)-one (9CI), KB-254121, A22248
InChIKey: KHRZFVYHKRMYLE-UHFFFAOYSA-N | ||||||||
• FURO[2,3-C]PYRIDIN-3(2H)-ONE HYDROCHLORIDE
IUPAC Name: furo[2,3-c]pyridin-3-one;hydrochloride | CAS Registry Number: 106531-51-5 Synonyms: Furo[2,3-c]pyridin-3(2H)-one hydrochloride, SureCN3597821, KB-254122
InChIKey: FWVRHCYASFZWGO-UHFFFAOYSA-N | ||||||||
• FURO[3,2-B]PYRIDIN-3(2H)-ONE
IUPAC Name: furo[3,2-b]pyridin-3-one | CAS Registry Number: 119293-03-7 Synonyms: furo[3,2-b]pyridin-3(2H)-one, ACMC-20moa7, furo[4,5-b]pyridin-3-one, SCHEMBL4507981, CTK0H3171, PBITTYWTCTZBSX-UHFFFAOYSA-N, AKOS023833178, ZINC100089873, FCH1187044, QC-1127, SC-87703, AB0088768
InChIKey: PBITTYWTCTZBSX-UHFFFAOYSA-N | ||||||||
• Gabexate Mesylate
IUPAC Name: [N'-[6-(4-ethoxycarbonylphenoxy)-6-oxohexyl]carbamimidoyl]azanium; methanesulfonate | CAS Registry Number: 56974-61-9 Synonyms: Gabexate mesilate, Gabexate mesylate, Gabexate monomethanesulfonate, Gabexato mesilato [Spanish], C16H23N3O4.CH4O3S, LS-35906, Ethyl p-(6-guanidinohexanoxyloxy)benzoate methanesulfonate, Ethyl p-(6-guanidinohexanoyloxy) benzoate methanesulfonate, p-Hydroxybenzoic acid ethyl ester 6-guanidinohexanoate mesilate, Benzoic acid, 4-((6-((aminoiminomethyl)amino)-1-oxohexyl)oxy)-, ethyl ester, monomethanesulfonate, FOY, BENZOIC ACID, 4-((6-((AMINOIMINOMETHYL)AMINO)-1-OXOHEXYL)OXY)-, ETHYL ESTER, MON, 39492-01-8, Benzoic acid, 4-((6-((aminoiminomethyl)amino)-1-oxohexyl)oxy)-, ethyl ester,monomethanesulfonate
InChIKey: DNTNDFLIKUKKOC-UHFFFAOYSA-N | ||||||||
• Ganetespib; STA-9090
IUPAC Name: (5Z)-5-(4-hydroxy-6-oxo-3-propan-2-ylcyclohexa-2,4-dien-1-ylidene)-4-(1-methylindol-5-yl)-1,2,4-triazolidin-3-one | CAS Registry Number: 888216-25-9 Synonyms: Ganetespib, STA9090, UNII-2E8412Y946, STA-9090, Ganetespib (USAN), Ganetespib,STA-9090, Ganetespib [USAN:INN], Ganetespib - STA-9090, CHEMBL2103879, QCR-148, BCP0726000115, 2E8412Y946, D10126, 3H-1,2,4-Triazol-3-one, 5-(2,4-dihydroxy-5-(1-methylethyl)phenyl)-2,4-dihydro-4-(1- methyl-1H-indol-5-yl)-, 5-(2,4-Dihydroxy-5-(1-methylethyl)phenyl)-4-(1-methyl-1H-indol-5-yl)-2,4-dihydro-3H- 1,2,4-triazol-3-one, 5-[2,4-Dihydroxy-5-(1-methylethyl)phenyl]-2,4-dihydro-4-(1-methyl-1H-indol-5-yl)-3H-1,2,4-triazol-3-one, 5-[2,4-Dihydroxy-5-(Propan-2-Yl)phenyl]-4-(1-Methyl-1h-Indol-5-Yl)-2,4-Dihydro-3h-1,2,4-Triazol-3-One, TUH
InChIKey: MWTUOSWPJOUADP-XDJHFCHBSA-N | ||||||||
• GDC-0032
IUPAC Name: 2-methyl-2-[4-[2-(5-methyl-2-propan-2-yl-1,2,4-triazol-3-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl]pyrazol-1-yl]propanamide | CAS Registry Number: 1282512-48-4 Synonyms: CHEMBL2387080, Taselisib, Taselisib [INN], SureCN1485247, UNII-L08J2O299M, KB-145919, S7103,GDC0032,RG7604,1282512-48-4
InChIKey: BEUQXVWXFDOSAQ-UHFFFAOYSA-N | ||||||||
• GDC-0068
IUPAC Name: (2S)-2-(4-chlorophenyl)-1-[4-[(5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl]piperazin-1-yl]-3-(propan-2-ylamino)propan-1-one | CAS Registry Number: 1001264-89-6 Synonyms: CHEMBL2177390, GDC 0068, Ipatasertib, RG 7440, SureCN191659, cc-616, GDC0068, BCP9000712, CS-0975, RG-7440, GDC-0068 (RG7440), NCGC00346714-01, HY-15186, QC-10488, BCP0726000195, GDC-0068|1001264-89-6|GDC0068|GDC 0068|RG-7440, (2s)-2-(4-Chlorophenyl)-1-{4-[(5r,7r)-7-Hydroxy-5-Methyl-6,7-Dihydro-5h-Cyclopenta[d]pyrimidin-4-Yl]piperazin-1-Yl}-3-(Propan-2-Ylamino)propan-1-One, 0RF
InChIKey: GRZXWCHAXNAUHY-NSISKUIASA-N | ||||||||
• GDC-0349
IUPAC Name: 1-ethyl-3-[4-[4-[(3S)-3-methylmorpholin-4-yl]-7-(oxetan-3-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-2-yl]phenyl]urea | CAS Registry Number: 1207360-89-1 Synonyms: CHEMBL2331680, SureCN1831520, GDC0349, UNII-579255I6O9, CS-0700, HY-15248, GDC-0349|1207360-89-1|GDC0349
InChIKey: RGJOJUGRHPQXGF-INIZCTEOSA-N | ||||||||
• GDC0980
IUPAC Name: (2S)-1-[4-[[2-(2-aminopyrimidin-5-yl)-7-methyl-4-morpholin-4-ylthieno[3,2-d]pyrimidin-6-yl]methyl]piperazin-1-yl]-2-hydroxypropan-1-one | CAS Registry Number: 1032754-93-0 Synonyms: GDC-0980, Apitolisib, CHEMBL1922094, RG7422, 1032754-93-0, (2s)-1-(4-{[2-(2-Aminopyrimidin-5-Yl)-7-Methyl-4-(Morpholin-4-Yl)thieno[3,2-D]pyrimidin-6-Yl]methyl}piperazin-1-Yl)-2-Hydroxypropan-1-One, (S)-1-(4-((2-(2-aminopyrimidin-5-yl)-7-methyl-4-morpholinothieno[3,2-d]pyrimidin-6-yl)methyl)piperazin-1-yl)-2-hydroxypropan-1-one, GNE 390; GDC 0980; RG 7422, GDC 0980, PubChem24448, cc-6, Apitolisib [USAN:INN], SureCN466297, UNII-1C854K1MIJ, QCR-182, GDC-0980,RG7422, RG7422, BCP9000717, CS-0590, GDC-0980.1, RG 7422
InChIKey: YOVVNQKCSKSHKT-HNNXBMFYSA-N | ||||||||
• Gefitinib
IUPAC Name: N-(3-chloro-4-fluorophenyl)-7-methoxy-6-(3-morpholin-4-ylpropoxy)quinazolin-4-amine | CAS Registry Number: 184475-35-2 Synonyms: Iressa, Irressat, Gefitini; Iressa, Gefitinib [USAN], Iressa (TN), nchembio866-comp14, nchembio.117-comp18, ZD1839, KBioSS_002241, Gefitinib (JAN/USAN/INN), ZD 1839, CCRIS 9011, STOCK6S-52331, CHEBI:49668, ZD-1839, CID123631, NSC715055, DB00317, NCGC00159455-02, NCGC00159455-03
InChIKey: XGALLCVXEZPNRQ-UHFFFAOYSA-N | ||||||||
• Geldanamycin
IUPAC Name: [(3R,5S,6R,7S,8E,10S,11S,12Z,14E)-6-hydroxy-5,11,21-trimethoxy-3,7,9,15-tetramethyl-16,20,22-trioxo-17-azabicyclo[16.3.1]docosa-1(21),8,12,14,18-pentaen-10-yl] carbamate | CAS Registry Number: 30562-34-6 Synonyms: geldanamycin, geldanomycin, Geldanamycin (9CI), nchembio.83-comp18, BODIPY-labeled Geldanamycin, BSPBio_001073, NChemBio.2007.10-comp1, CID5288382, IDI1_002122, NCGC00163449-01, NCGC00163449-02, Geldanamycin, Streptomyces hygroscopicus, A00271, C11222, U-29135, 2-Azabicyclo[16.3.1]docosane, geldanamycin deriv., GDM, (4E,6Z,8S,9S,10E,12S,13R,14S,16R)-13-hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl carbamate, [(3R,5S,6R,7S,8E,10S,11S,12Z,14E)-6-hydroxy-5,11,21-trimethoxy-3,7,9,15-tetramethyl-16,20,22-trioxo-17-azabicyclo[16.3.1]docosa-1(21),8,12,14,18-pentaen-10-yl] carbamate, [(3S,5S,6R,7S,8E,10R,11S,12Z,14E)-6-Hydroxy-5,11,21-trimethoxy-3,7,9,15-tetramethyl-16,20,22-trioxo-17-azabicyclo[16.3.1]docosa-8,12,14,18,21-pentaen-10-yl] carbamate
InChIKey: QTQAWLPCGQOSGP-KSRBKZBZSA-N | ||||||||
• Gemcitabine HCL
IUPAC Name: 4-amino-1-[(2R,4R,5R)-3,3-difluoro-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]pyrimidin-2-one hydrochloride | CAS Registry Number: 122111-03-9 Synonyms: Gemzar, Gemzar (TN), GEMCITABINE HYDROCHLORIDE, Ambap6387, LY188011 hydrochloride, Gemcitabine HCL (Gemzar), C9H11F2N3O4.HCl, Gemcitabine hydrochloride [USAN], Gemcitabine hydrochloride (JAN/USAN), 2',2'-Difluorodeoxycytidine monohydrochloride, CPD000469146, LS-59069, SAM001246550, TL8000589, 2'-Deoxy-2',2'-difluorocytidine monohydrochloride, D01155, Cytidine, 2'-deoxy-2',2'-difluoro-, monohydrochloride, 2'-Deoxy-2',2'-difluorocytidine monohydrochloride (beta-isomer), 103882-84-4, 95058-81-4
InChIKey: OKKDEIYWILRZIA-OSZBKLCCSA-N | ||||||||
• Genistein
IUPAC Name: 5,7-dihydroxy-3-(4-hydroxyphenyl)chromen-4-one | CAS Registry Number: 446-72-0 Synonyms: genistein, Genisteol, Genisterin, Prunetol, Sophoricol, Genestein, Differenol A, Isoflavone, Bonistein, 4',5,7-Trihydroxyisoflavone, 5,7,4'-Trihydroxyisoflavone, Lactoferrin-genistein, nchembio.76-comp6, Spectrum_000320, Tocris-1110, 1x7r, SpecPlus_000305, Spectrum2_000638, Spectrum3_000678, Spectrum4_001543
InChIKey: TZBJGXHYKVUXJN-UHFFFAOYSA-N | ||||||||
• Glimepiride
IUPAC Name: 4-ethyl-3-methyl-N-[2-[4-[(4-methylcyclohexyl)carbamoylsulfamoyl]phenyl]ethyl]-5-oxo-2H-pyrrole-1-carboxamide | CAS Registry Number: 93479-97-1 Synonyms: glimepiride, Amaryl, Glimepirid, Amarel, Glimepride, Endial, Glimepirida, Glimepiridum, Glymepirid, Avandaryl, Duetact, Glimer, Roname, Solosa, Mixture Name, Glimepiridum [Latin], Glimepirida [Spanish], Amaryl (TN), Hoe-490, Prestwick0_000651
InChIKey: WIGIZIANZCJQQY-UHFFFAOYSA-N | ||||||||
• GNF-2
IUPAC Name: 3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]benzamide | CAS Registry Number: 778270-11-4 Synonyms: Bcr-abl Inhibitor, GNF2, (3-(6)-(4-Trifluoromethoxy-phenylamino)-pyrimidin-4-yl)-benzamide, 3-[6-[[4-(Trifluoromethoxy)phenyl]amino]-4-pyrimidinyl]benzamide, SMR000463555, 3-(6-{[4-(Trifluoromethoxy)phenyl]amino}pyrimidin-4-Yl)benzamide, 3-[6-[[4-(trifluoromethoxy)phenyl]amino]pyrimidin-4-yl]benzamide, 3k5v, AC1NSKR6, SureCN925002, AC1Q4ZE7, UNII-6D7Q9Z2W7T, cc-647, MLS000911539, MLS003105943, G9420_SIGMA, CHEMBL483847, QCR-247, CHEBI:585249, HMS2043N17
InChIKey: WEVYNIUIFUYDGI-UHFFFAOYSA-N | ||||||||
• GO 6983; 3-[1-[3-(DIMETHYLAMINO)PROPYL]-5-METHOXY-1H-INDOL-3-YL]- 4-(1H-INDOL-3-YL)-1H-PYRROLE-2,5-DIONE
IUPAC Name: 3-[1-[3-(dimethylamino)propyl]-5-methoxyindol-3-yl]-4-(1H-indol-3-yl)pyrrole-2,5-dione | CAS Registry Number: 133053-19-7 Synonyms: go 6983, Gö 6983, 2-(1-(3-dimethylaminopropyl)-5-methoxyindol-3-yl)-3-(1h-indol-3-yl)maleimide, 2-[1-(3-Dimethylaminopropyl)-5-methoxyindol-3-yl]-3-(1H-indol-3-yl) maleimide, 3-[1-[3-(Dimethylamino)propyl]-5-methoxy-1H-indol-3-yl]-4-(1H-indol-3-yl)-1H-pyrrole-2,5-dione, AC1L1G2N, AC1Q6P6S, SureCN1680253, G1918_SIGMA, Goe 6983, CHEMBL261491, CTK4B8320, MolPort-003-941-462, HMS3229E15, Go-6893, AR-1C5949, IN1307, AG-K-40753, CCG-206756, NCGC00163505-01
InChIKey: LLJJDLHGZUOMQP-UHFFFAOYSA-N | ||||||||
• Griseofulvin
IUPAC Name: (2S,5'R)-7-chloro-3',4,6-trimethoxy-5'-methylspiro[1-benzofuran-2,4'-cyclohex-2-ene]-1',3-dione | CAS Registry Number: 126-07-8 Synonyms: griseofulvin, Fulvicin, Amudane, Delmofulvina, Griscofulvin, Griseofulvinum, Grizeofulvin, Fulvistatin, Grisefuline, Grisofulvin, Spirofulvin, Fulvinil, Fungivin, Gresfeed, Grifulin, Grifulvin, Grisactin, Griseomix, Grisetin, Grisovin
InChIKey: DDUHZTYCFQRHIY-RBHXEPJQSA-N | ||||||||
• GSK 1363089
IUPAC Name: 1-N'-[3-fluoro-4-[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyphenyl]-1-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | CAS Registry Number: 849217-64-7 Synonyms: Foretinib, XL880, GSK089, GSK1363089, EXEL-2880, XL-880, S1111_Selleck, GSK1363089G, XL 880, GSK-1363089, CHEMBL1230609, Foretinib (XL-880), GSK089, EXEL-2880, 849217-64-7, GSK1363089, GSK089, foretinib, EXEL-2880, XL880, 88Z, 937176-80-2, N-[3-Fluoro-4-[[6-methoxy-7-[3-(4-morpholinyl)propoxy]-4-quinolinyl]oxy]phenyl]-N'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide, EXEL 2880, n-(3-fluoro-4-((6-methoxy-7-(3-(4-morpholinyl)propoxy)-4-quinolinyl)oxy)phenyl)-n'-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide, PubChem22993
InChIKey: CXQHYVUVSFXTMY-UHFFFAOYSA-N | ||||||||
• GSK 2126458
IUPAC Name: 2,4-difluoro-N-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamide | CAS Registry Number: 1086062-66-9 Synonyms: GSK2126458, GSK-2126458, 2,4-Difluoro-N-[2-methoxy-5-[4-(4-pyridazinyl)-6-quinolinyl]-3-pyridinyl]benzenesulfonamide, 2,4-difluoro-N-(2-methoxy-5-(4-(pyridazin-4-yl)quinolin-6-yl)pyridin-3-yl)benzenesulfonamide, GSK212, GSK 212, GSK-212, 2,4-difluoro-N-{2-methoxy-5-[4-(pyridazin-4-yl)quinolin-6-yl]pyridin-3-yl}benzenesulfonamide, PubChem22430, cc-65, SureCN623194, UNII-1X8F5A3NA0, GSK-458, 3l08, ABP000103, AKOS015904655, CS-0085, QC-7243, RL00368, NCGC00250408-01
InChIKey: CGBJSGAELGCMKE-UHFFFAOYSA-N | ||||||||
• GSK 2334470
IUPAC Name: (3S,6R)-1-[6-(3-amino-1H-indazol-6-yl)-2-(methylamino)pyrimidin-4-yl]-N-cyclohexyl-6-methylpiperidine-3-carboxamide | CAS Registry Number: 1227911-45-6 Synonyms: GSK2334470, SureCN1317022, CHEMBL1765740, CHEBI:1240766, CS-0917, QC-8425, GSK-2334470, HY-14981, KB-77621, GSK2334470|1227911-45-6|GSK-2334470, (3S,6R)-1-(6-(3-amino-1H-indazol-6-yl)-2-(methylamino)pyrimidin-4-yl)-N-cyclohexyl-6-methylpiperidine-3-carboxamide
InChIKey: QLPHOXTXAKOFMU-WBVHZDCISA-N | ||||||||
• GSK 525762A
IUPAC Name: 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide | CAS Registry Number: 1260907-17-2 Synonyms: CHEMBL1232461, 2-[(4s)-6-(4-Chlorophenyl)-8-Methoxy-1-Methyl-4h-[1,2,4]triazolo[4,3-A][1,4]benzodiazepin-4-Yl]-N-Ethylacetamide, EAM, 3p5o, SureCN1872390, GSK525762A, GSK-525762A, CCG-208698, CS-0717, NCGC00263621-02, HY-13032, GSK 525762A|1260907-17-2|GSK-525762A
InChIKey: AAAQFGUYHFJNHI-SFHVURJKSA-N | ||||||||
• GSK 690693
IUPAC Name: 4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[[(3S)-piperidin-3-yl]methoxy]imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | CAS Registry Number: 937174-76-0 Synonyms: GSK690693, GSK-690693, (S)-4-(2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-(piperidin-3-ylmethoxy)-1H-imidazo[4,5-c]pyridin-4-yl)-2-methylbut-3-yn-2-ol, GSK 690693, GSK-690693, 937174-76-0, cc-44, SureCN310452, UNII-GWH480321B, CHEMBL494089, CTK5H2854, ABP000406, ANW-64913, DNC008950, AKOS015904356, AG-L-59959, BCP9000745, QC-7252, NCGC00263181-01, AK103308, HY-10249, KB-77630
InChIKey: KGPGFQWBCSZGEL-ZDUSSCGKSA-N | ||||||||
• GSK J4
IUPAC Name: ethyl 3-[[2-pyridin-2-yl-6-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)pyrimidin-4-yl]amino]propanoate | CAS Registry Number: 1373423-53-0 Synonyms: GSK-J4, KB-145933, BRD-K98203492-001-01-1
InChIKey: WBKCKEHGXNWYMO-UHFFFAOYSA-N | ||||||||
• GSK-1120212
IUPAC Name: N-[3-[3-cyclopropyl-5-(2-fluoro-4-iodoanilino)-6,8-dimethyl-2,4,7-trioxopyrido[4,3-d]pyrimidin-1-yl]phenyl]acetamide | CAS Registry Number: 871700-17-3 Synonyms: Trametinib, GSK1120212, GSK 1120212, Mekinist, JTP-74057, JTP 74057, UNII-33E86K87QN, CHEBI:75998, JTP74057, N-[3-[3-Cyclopropyl-5-[(2-fluoro-4-iodophenyl)amino]-3,4,6,7-tetrahydro-6,8-dimethyl-2,4,7-trioxopyrido[4,3-d]pyrimidin-1(2H)-yl]phenyl]acetamide, JTP-74057, 871700-17-3, trametinibum, N-(3-(3-Cyclopropyl-5-((2-fluoro-4-iodophenyl)amino)-6,8-dimethyl-2,4,7-trioxo-3,4,6,7- tetrahydropyrido(4,3-d)pyrimidin-1(2H)-yl)phenyl)acetamide, N-(3-{3-cyclopropyl-5-((2-fluoro-4-iodophenyl)amino)-6,8-dimethyl-2,4,7-trioxo-3,4,6,7- tetrahydropyrido(4,3-d)pyrimidin-1(2H)-yl}phenyl)acetamide, Trametinib (USAN), Trametinib [USAN:INN], cc-37, SureCN170938, QCR-39, Trametinib (GSK1120212)
InChIKey: LIRYPHYGHXZJBZ-UHFFFAOYSA-N | ||||||||
• GSK-2636771
IUPAC Name: 2-methyl-1-[[2-methyl-3-(trifluoromethyl)phenyl]methyl]-6-morpholin-4-ylbenzimidazole-4-carboxylic acid | CAS Registry Number: 1372540-25-4 Synonyms: GSK2636771, UNII-DW94IAT0LS, SureCN1280998, cc-414, QCR-187, BCP9000741, CS-0747, NCGC00345796-01, HY-15245, GSK2636771|1372540-25-4|GSK-2636771, S8002, GSK 2636771, GSK-2636771, 1372540-25-4, 2-Methyl-1-((2-methyl-3-(trifluoromethyl)phenyl)methyl)-6-(4-morpholinyl)-1H-benzimidazole-4-carboxylic acid, 2-Methyl-1-((2-methyl-3-(trifluoromethyl)phenyl)methyl)-6-morpholino-benzimidazole-4-carboxylic acid, 2-methyl-1-(2-methyl-3-(trifluoromethyl)benzyl)-6-morpholino-1H-benzo[d]imidazole-4-carboxylic acid
InChIKey: XTKLTGBKIDQGQL-UHFFFAOYSA-N | ||||||||
• GSK-3BETA INHIBITOR XII
IUPAC Name: 3-[[6-(3-aminophenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]oxy]phenol | CAS Registry Number: 601514-19-6 Synonyms: TWS119, TWS 119, TWS-119, GSK-3beta Inhibitor XII, TWS119, Neurogenesis Inducer, TWS119, 3-(6-(3-aminophenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yloxy)phenol, 3-[[6-(3-Aminophenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]oxy]phenol, 3-{[6-(3-aminophenyl)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]oxy}phenol, 3-((6-(3-AMINOPHENYL)-7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)OXY)PHENOL, GSK inhibitor XII, S1590_Sselleck, K00245, SureCN5559045, cc-510, CHEMBL405759, CTK8F1085, CHEBI:530386, MolPort-003-791-493, BCPP000029, HMS3229M16
InChIKey: VPVLEBIVXZSOMQ-UHFFFAOYSA-N | ||||||||
• GSK1210151A (I-BET151)
IUPAC Name: 7-(3,5-dimethyl-1,2-oxazol-4-yl)-8-methoxy-1-[(1R)-1-pyridin-2-ylethyl]-3H-imidazo[4,5-c]quinolin-2-one | CAS Registry Number: 1300031-49-5 Synonyms: CHEMBL2017291, GSK1210151A, 7-(3,5-Dimethyl-4-isoxazolyl)-1,3-dihydro-8-methoxy-1-[(1R)-1-(2-pyridinyl)ethyl]-2H-imidazo[4,5-c]quinolin-2-one, 3zyu, 4alg, 1GH, 7-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-8-Methoxy-1-[(1r)-1-(Pyridin-2-Yl)ethyl]-1h,2h,3h-Imidazo[4,5-C]quinolin-2-One, SureCN1906755, cc-415, I-BET151, I-BET 151, QCR-236, GSK 1210151A, GSK-1210151A, AKOS016004407, BCP9000734, CS-0930, RL01425, GSK1210151A/I-BET 151, NCGC00344588-01
InChIKey: VUVUVNZRUGEAHB-CYBMUJFWSA-N | ||||||||
• GSK1838705A
IUPAC Name: 2-[[2-[[1-[2-(dimethylamino)acetyl]-5-methoxy-2,3-dihydroindol-6-yl]amino]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino]-6-fluoro-N-methylbenzamide | CAS Registry Number: 1116235-97-2 Synonyms: GSK-1838705A, SureCN2205605, SureCN12428872, cc-268, CHEMBL464552, BCP9000736, CS-0695, pyrrolo[2,3-d]pyrimidine deriv., 40, RL00469, NCGC00346647-01, HY-13020, X7516, GSK1838705A|1116235-97-2|GSK-1838705A, 2-((2-((1-((dimethylamino)ethanoyl)-5-(methyloxy)-2,3-dihydro-1h-indol-6-yl)amino)-7h-pyrrolo(2,3-d)pyrimidin-4-yl)amino)-6-fluoro-n-methylbenzamide, 2-(2-(1-(2-(dimethylamino)acetyl)-5-methoxyindolin-6-ylamino)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-6-fluoro-N-methylbenzamide, 2-{[2-({1-[2-(dimethylamino)acetyl]-5-methoxy-2,3-dihydroindol-6-yl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}-6-fluoro-N-methylbenzamide
InChIKey: HZTYDQRUAWIZRE-UHFFFAOYSA-N | ||||||||
• GSK1904529A
IUPAC Name: N-(2,6-difluorophenyl)-5-[3-[2-[5-ethyl-2-methoxy-4-[4-(4-methylsulfonylpiperazin-1-yl)piperidin-1-yl]anilino]pyrimidin-4-yl]imidazo[1,2-a]pyridin-2-yl]-2-methoxybenzamide | CAS Registry Number: 1089283-49-7 Synonyms: GSK 1904529A, N-(2,6-Difluorophenyl)-5-[3-[2-[[5-ethyl-2-(methyloxy)-4-[4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl]phenyl]amino]-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl]-2-(methyloxy)benzamide, S1093_Selleck, PubChem22431, cc-35, SureCN309890, CHEMBL466397, CHEBI:575598, ABP000158, GSK-1904529A, EX-8674, QC-7246, RL00381, NCGC00253439-01, HY-10524, KB-77619, GSK1904529A-Supplied by Selleck Chemicals, Y0282, GSK 1904529A (GSK 4529), A24618
InChIKey: MOSKATHMXWSZTQ-UHFFFAOYSA-N | ||||||||
• GSK343
IUPAC Name: N-[(6-methyl-2-oxo-4-propyl-1H-pyridin-3-yl)methyl]-6-[2-(4-methylpiperazin-1-yl)pyridin-4-yl]-1-propan-2-ylindazole-4-carboxamide | CAS Registry Number: 1346704-33-3 Synonyms: CHEMBL2204995, SureCN14716863, KB-145929
InChIKey: ULNXAWLQFZMIHX-UHFFFAOYSA-N |